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H-7.Dihydrochloride

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产品名称: H-7.Dihydrochloride
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简单介绍

CAS:108930-17-2Formula:C14H17N3O2S.2HClMW:291.4.73.0Appearance:WhitetoLightYellowSolidPurity:>98%


H-7.Dihydrochloride  的详细介绍

Potent inhibitor of PKA (Ki=3.0 μm), PKC (Ki=6 μm), PKG (Ki=5.8 nM), and myosin light chain kinase (Ki=97 μm). Selectivity for PKC can achieved when used in conjunction with HA-1004.

Attached is a published reference from researchers who have used our H-7.Dihydrochloride product.

  • EXPERIMENTAL AND MOLECULAR MEDICINE/ONCOLOGY/PATHOLOGY: Polyenoic Fatty Acid Ratios Alter Fibroblast Collagen Production Via PGE2 and PGE Receptor Subtype Response, Yi Jia and John J. Turek, Exp Biol Med, Jul 2004; 229: 676 - 683.

Additional Information

Product #H-1020
CAS #108930-17-2
Chemical Name(1-(5-isoquinolinesulfonyl)-2-methylpiperazine.2HCl)
FormulaC14H17N3O2S.2HCl
MW291.4 . 73.0
AppearanceWhite to Light Yellow Solid
Purity>98%
SolubilitySoluble in Water.
Storage Temp-20°C

Additional Information

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